TAR-200 for Bacillus Calmette-Guérin–Unresponsive High-Risk Non–Muscle-Invasive Bladder Cancer: Results From the Phase IIb SunRISe-1 Study

M Michiel S. Van Der Heijden (Department of Medical Oncology Netherlands Cancer Institute Amsterdam Netherlands) J Joseph M. Jacob (Department of Urology, SUNY Upstate Medical University, Syracuse, NY) F Félix Guerrero-Ramos C Christopher M. Pieczonka (Clinical Research, U.S. Urology Partners and Associated Medical Professionals of New York, Syracuse) P Philipp Spiegelhalder (Urologie Neandertal, Gemeinschaftspraxis für Urologie, Mettmann, Germany) K Katie S. Murray (Department of Urology, NYU Grossman School of Medicine, New York, NY) K Katharine Stromberg (Johnson & Johnson, Raritan, NJ) J Jason Martin A Abhijit Shukla (Johnson & Johnson, Lexington, MA) C Christopher J. Cutie (Johnson & Johnson, Lexington, MA) K Kristi Bertzos (Johnson & Johnson, Horsham, PA) S Shalaka Hampras (Johnson & Johnson, Raritan, NJ) H Hussein Sweiti (Johnson & Johnson, Spring House, PA) M Manish Patel T Thierry Roumeguere C Charles Van Praet H Harm Arentsen B Bart De Troyer (Department of Urology, VITAZ, Sint-Niklaas, Belgium) F Frederic Baekelandt K Karel Decaestecker G Girish Kulkarni W Wassim Kassouf G George Vrabec S Sabrina Falkowski (Clinique François Chénieux, Limoges, France) G Geraldine Pignot (Institut Paoli-Calmettes, Department of Surgical Oncology, Marseille, France) E Evanguelos Xylinas (Department of Urology, Bichat-Claude Bernard Hospital, Assistance Publique-Hôpitaux de Paris, Université de Paris Cité, Paris, France) M Morgan Roupret (Sorbonne Université, Pitié-Salpêtrière Hospital, AP-HP, Paris, France) M Marc Colombel R Romain Mathieu (University of Rennes Hospital Centre, Department of Urology, Rennes, France) B Benoit Wolff M Marc-Olivier Timsit X Xavier Artignan (Hôpital Saint Grégoire, Rennes, France) S Stephane Droupy H Herve Lang M Mathieu Roumiguié (Institut Universitaire du Cancer Toulouse Oncopole CHU, Toulouse, France) F Frank Bladou C Catherine Becht M Martin Bögemann (Department of Urology, Münster University Hospital, Münster, Germany) P Phillipp Spiegelhalder J Jorg Klier T Tilman Toderhofer E Eva Hellmis P Petros Sountoulides K Konstantinos Hatzimouratidis G Giuseppe Simone (Department of Urology, 'Regina Elena' National Cancer Institute, Rome, Italy) L Luca Galli F Frederico Deho A Andrea Minervini A Andrea Necchi (Department of Medical Oncology Fondazione IRCCS Istituto Nazionale dei Tumori University of Milan Milan Italy) T Takashi Kawahara S Shuya Kandori M Masao Tsujihata S Shinji Urakami T Taek Won Kang (Department of Urology, Chonnam National University Medical School, Gwangju, Republic of Korea) J Ja Hyeon Ku (Seoul National University Hospital, Seoul, South Korea) K Kang Su Cho (Department of Urology, Gangnam Severance Hospital, Yonsei University College of Medicine, Seoul, South Korea) W Wonho Jung (C1 Gas Refinery Research and Development Center, Sogang University) H Ho Kyung Seo (Center for Urologic Cancer, National Cancer Center, Goyang, Korea, Republic of) J Jong Kil Nam (Department of Urology, Pusan National University Yangan Hospital, Pusan National University School of Medicine, Yangsan, South Korea) D Diederik Somford M Michiel Van der Heijden A Antonio Morais V Vania Grenha J Jorge Rebola S Sandra Custodio V Vagif Atduev (Volga District Medical Center, Federal Medical-Biological Agency, Nizhny Novgorod, Russian Federation) D Denis Kholtdobin J Jose Luis Alvarez-Ossorio Fernandez J Javier Romero Otero F Felix Guerrero Ramos B Bernardo Herrera Imbroda (Urology Department, Hospital Universitario Virgen de la Victoria, IBIMA-Plataforma Bionand, Málaga, Malaga, Spain) P Pol Servian Vives N Nelson Canales Casco (Hospital de Jerez de la Frontera y Punta Europa, Cádiz, Spain) M Mario Eduardo Alvarez Maestro D David Morris (Dayton Children’s Hospital, Dayton, OH) S Siamak Daneshmand (Department of Urology, Keck School of Medicine of University of Southern California, Norris Comprehensive Cancer Center) C Curtis Dunshee D Daniel Zainfeld (Urology San Antonio, San Antonio, TX) K Katie Murray L Laurence Belkoff (Midlantic Urology, Bala Cynwyd, PA) P Peter Earl Clark Y Yair Lotan (Department of Urology, UT Southwestern Medical Center, Dallas, TX) J Joseph Jacob D David Cahn (Colorado Urology, Lakewood, CO) C Christopher Pieczonka A Amy Luckenbaugh (Vanderbilt University Medical Center, Nashville, TN) M Marc Pliskin J Jason Hafron (Corewell Health William Beaumont University Hospital, Royal Oak, MI) E Eugene Cone (Urology of Indiana, Greenwood, IN) B Brian Mazzarella (Urology Austin, Austin, TX) R Richard David

Abstract

PURPOSE TAR-200 is a first-in-class intravesical drug-releasing system designed to provide sustained delivery of gemcitabine in the bladder. TAR-200 alone or in combination with cetrelimab (PD-1 inhibitor) could improve outcomes in patients with bacillus Calmette-Guérin (BCG)–unresponsive high-risk non–muscle-invasive bladder cancer (NMIBC) ineligible for or refusing radical cystectomy. METHODS In this phase IIb parallel cohort study, patients with BCG-unresponsive carcinoma in situ (CIS) with/without papillary disease received TAR-200 monotherapy (Cohort 2 [C2]), TAR-200 plus cetrelimab (C1), or cetrelimab monotherapy (C3). Patients with BCG-unresponsive high-risk papillary disease–only NMIBC received TAR-200 monotherapy (C4). TAR-200 was dosed through month 24 and cetrelimab through month 18. Primary end points were centrally confirmed overall complete response (CR) rate (C1-3) or disease-free survival (DFS) rate (C4) (ClinicalTrials.gov number: NCT04640623 ). RESULTS At data cutoff (March 31, 2025), 53, 85, 28, and 52 patients were treated in C1-4, respectively. In C2, CR rate and median duration of response were 82.4% (95% CI, 72.6 to 89.8) and 25.8 months (95% CI, 8.3 to not estimable), respectively. In C4, 6-, 9-, and 12-month DFS rates were 85.3% (95% CI, 71.6 to 92.7), 81.1% (95% CI, 66.7 to 89.7), and 70.2% (95% CI, 51.6 to 82.8), respectively. In C1 and C3, CR rates were 67.9% (95% CI, 53.7 to 80.1) and 46.4% (95% CI, 27.5 to 66.1), respectively. Rates of grade ≥3 treatment-related adverse events (AEs) were 12.9%, 13.5%, 37.7%, and 7.1% in C2, C4, C1, and C3, respectively, and of serious treatment-related AEs, 5.9%, 5.8%, 15.1%, and 3.6%. No treatment-related deaths occurred. CONCLUSION TAR-200 monotherapy was well tolerated, with a high CR rate, durable responses, and prolonged DFS in patients with BCG-unresponsive high-risk NMIBC. TAR-200 monotherapy offered a more favorable risk-benefit profile versus TAR-200 plus cetrelimab or cetrelimab alone in BCG-unresponsive CIS.

Article Details

Volume / Issue Vol. 43, Issue 33
Published November 20, 2025
Pages 3578-3588
ISSN 0732-183X
Publisher Lippincott Williams & Wilkins

Journal Info

Journal of Clinical Oncology

Lippincott Williams & Wilkins

ISSN: 0732-183X Health Sciences

Authors (91)

M

Michiel S. Van Der Heijden

Department of Medical Oncology Netherlands Cancer Institute Amsterdam Netherlands

J

Joseph M. Jacob

Department of Urology, SUNY Upstate Medical University, Syracuse, NY

F

Félix Guerrero-Ramos

C

Christopher M. Pieczonka

Clinical Research, U.S. Urology Partners and Associated Medical Professionals of New York, Syracuse

P

Philipp Spiegelhalder

Urologie Neandertal, Gemeinschaftspraxis für Urologie, Mettmann, Germany

K

Katie S. Murray

Department of Urology, NYU Grossman School of Medicine, New York, NY

K

Katharine Stromberg

Johnson & Johnson, Raritan, NJ

J

Jason Martin

A

Abhijit Shukla

Johnson & Johnson, Lexington, MA

C

Christopher J. Cutie

Johnson & Johnson, Lexington, MA

K

Kristi Bertzos

Johnson & Johnson, Horsham, PA

S

Shalaka Hampras

Johnson & Johnson, Raritan, NJ

H

Hussein Sweiti

Johnson & Johnson, Spring House, PA

M

Manish Patel

T

Thierry Roumeguere

C

Charles Van Praet

H

Harm Arentsen

B

Bart De Troyer

Department of Urology, VITAZ, Sint-Niklaas, Belgium

F

Frederic Baekelandt

K

Karel Decaestecker

G

Girish Kulkarni

W

Wassim Kassouf

G

George Vrabec

S

Sabrina Falkowski

Clinique François Chénieux, Limoges, France

G

Geraldine Pignot

Institut Paoli-Calmettes, Department of Surgical Oncology, Marseille, France

E

Evanguelos Xylinas

Department of Urology, Bichat-Claude Bernard Hospital, Assistance Publique-Hôpitaux de Paris, Université de Paris Cité, Paris, France

M

Morgan Roupret

Sorbonne Université, Pitié-Salpêtrière Hospital, AP-HP, Paris, France

M

Marc Colombel

R

Romain Mathieu

University of Rennes Hospital Centre, Department of Urology, Rennes, France

B

Benoit Wolff

M

Marc-Olivier Timsit

X

Xavier Artignan

Hôpital Saint Grégoire, Rennes, France

S

Stephane Droupy

H

Herve Lang

M

Mathieu Roumiguié

Institut Universitaire du Cancer Toulouse Oncopole CHU, Toulouse, France

F

Frank Bladou

C

Catherine Becht

M

Martin Bögemann

Department of Urology, Münster University Hospital, Münster, Germany

P

Phillipp Spiegelhalder

J

Jorg Klier

T

Tilman Toderhofer

E

Eva Hellmis

P

Petros Sountoulides

K

Konstantinos Hatzimouratidis

G

Giuseppe Simone

Department of Urology, 'Regina Elena' National Cancer Institute, Rome, Italy

L

Luca Galli

F

Frederico Deho

A

Andrea Minervini

A

Andrea Necchi

Department of Medical Oncology Fondazione IRCCS Istituto Nazionale dei Tumori University of Milan Milan Italy

T

Takashi Kawahara

S

Shuya Kandori

M

Masao Tsujihata

S

Shinji Urakami

T

Taek Won Kang

Department of Urology, Chonnam National University Medical School, Gwangju, Republic of Korea

J

Ja Hyeon Ku

Seoul National University Hospital, Seoul, South Korea

K

Kang Su Cho

Department of Urology, Gangnam Severance Hospital, Yonsei University College of Medicine, Seoul, South Korea

W

Wonho Jung

C1 Gas Refinery Research and Development Center, Sogang University

H

Ho Kyung Seo

Center for Urologic Cancer, National Cancer Center, Goyang, Korea, Republic of

J

Jong Kil Nam

Department of Urology, Pusan National University Yangan Hospital, Pusan National University School of Medicine, Yangsan, South Korea

D

Diederik Somford

M

Michiel Van der Heijden

A

Antonio Morais

V

Vania Grenha

J

Jorge Rebola

S

Sandra Custodio

V

Vagif Atduev

Volga District Medical Center, Federal Medical-Biological Agency, Nizhny Novgorod, Russian Federation

D

Denis Kholtdobin

J

Jose Luis Alvarez-Ossorio Fernandez

J

Javier Romero Otero

F

Felix Guerrero Ramos

B

Bernardo Herrera Imbroda

Urology Department, Hospital Universitario Virgen de la Victoria, IBIMA-Plataforma Bionand, Málaga, Malaga, Spain

P

Pol Servian Vives

N

Nelson Canales Casco

Hospital de Jerez de la Frontera y Punta Europa, Cádiz, Spain

M

Mario Eduardo Alvarez Maestro

D

David Morris

Dayton Children’s Hospital, Dayton, OH

S

Siamak Daneshmand

Department of Urology, Keck School of Medicine of University of Southern California, Norris Comprehensive Cancer Center

C

Curtis Dunshee

D

Daniel Zainfeld

Urology San Antonio, San Antonio, TX

K

Katie Murray

L

Laurence Belkoff

Midlantic Urology, Bala Cynwyd, PA

P

Peter Earl Clark

Y

Yair Lotan

Department of Urology, UT Southwestern Medical Center, Dallas, TX

J

Joseph Jacob

D

David Cahn

Colorado Urology, Lakewood, CO

C

Christopher Pieczonka

A

Amy Luckenbaugh

Vanderbilt University Medical Center, Nashville, TN

M

Marc Pliskin

J

Jason Hafron

Corewell Health William Beaumont University Hospital, Royal Oak, MI

E

Eugene Cone

Urology of Indiana, Greenwood, IN

B

Brian Mazzarella

Urology Austin, Austin, TX

R

Richard David