Structure of a lasso peptide bound ETB receptor provides insights into the mechanism of GPCR inverse agonism

W Wataru Shihoya H Hiroaki Akasaka P Peter A. Jordan (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) A Anna Lechner (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) B Bethany K. Okada (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) G Gabriella Costa Machado da Cruz (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) F Fumiya K. Sano T Tatsuki Tanaka R Ryo Kawahara (Graduate School of Science, The University of Tokyo, 7-3-1 Hongo, Bunkyo-ku, Tokyo 113-0033, Japan) R Rajan Chaudhari (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) H Hiroko Masamune M Mark J. Burk (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) O Osamu Nureki

Article Details

Volume / Issue Vol. 16, Issue 1
Published April 22, 2025
ISSN 2041-1723
Publisher Nature Portfolio

Journal Info

Nature Communications

Nature Portfolio

ISSN: 2041-1723 Open Access Life Sciences

Authors (13)

W

Wataru Shihoya

H

Hiroaki Akasaka

P

Peter A. Jordan

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

A

Anna Lechner

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

B

Bethany K. Okada

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

G

Gabriella Costa Machado da Cruz

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

F

Fumiya K. Sano

T

Tatsuki Tanaka

R

Ryo Kawahara

Graduate School of Science, The University of Tokyo, 7-3-1 Hongo, Bunkyo-ku, Tokyo 113-0033, Japan

R

Rajan Chaudhari

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

H

Hiroko Masamune

M

Mark J. Burk

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

O

Osamu Nureki