Residue-Selective Inhibitors Discovery via Covalent DNA-Encoded Chemical Libraries with Diverse Warheads

X Xinyuan Wu (State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica) J Jiayi Pan R Rufeng Fan (State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica) Y Yiwei Zhang (State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica) C Chao Wang G Guoliang Wang (School of Chinese Materia Medica) J Jiaxiang Liu (State Key Laboratory of Drug Research) M Mengqing Cui (State Key Laboratory of Drug Research) J Jinfeng Yue (State Key Laboratory of Drug Research) R Rui Jin Z Zhiqiang Duan (State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica) M Mingyue Zheng L Lianghe Mei (Suzhou Institute of Materia Medica) L Lu Zhou (School of Pharmacy) M Minjia Tan (State Key Laboratory of Drug Research) J Jing Ai (State Key Laboratory of Drug Research) X Xiaojie Lu (State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica)

Article Details

Volume / Issue Vol. 147, Issue 18
Published May 07, 2025
Pages 15469-15481
ISSN 0002-7863
Publisher American Chemical Society

Journal Info

Journal of the American Chemical Society

American Chemical Society

ISSN: 0002-7863 Physical Sciences

Authors (17)

X

Xinyuan Wu

State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica

J

Jiayi Pan

R

Rufeng Fan

State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica

Y

Yiwei Zhang

State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica

C

Chao Wang

G

Guoliang Wang

School of Chinese Materia Medica

J

Jiaxiang Liu

State Key Laboratory of Drug Research

M

Mengqing Cui

State Key Laboratory of Drug Research

J

Jinfeng Yue

State Key Laboratory of Drug Research

R

Rui Jin

Z

Zhiqiang Duan

State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica

M

Mingyue Zheng

L

Lianghe Mei

Suzhou Institute of Materia Medica

L

Lu Zhou

School of Pharmacy

M

Minjia Tan

State Key Laboratory of Drug Research

J

Jing Ai

State Key Laboratory of Drug Research

X

Xiaojie Lu

State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica