Proteomic Ligandability Maps of Phosphorus(V) Stereoprobes Identify Covalent TLCD1 Inhibitors

H Hayden A. Sharma (Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States) M Michael Bielecki (Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States) M Meredith A. Holm (Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States) T Ty M. Thompson (Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States) Y Yue Yin J Jacob B. Cravatt (Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States) T Timothy B. Ware (Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States) A Alex Reed (Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States) M Molhm Nassir T Tamara El-Hayek Ewing (Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States) B Bruno Melillo J J. Fernando Bazan (ℏ Bioconsulting LLC) P Phil S. Baran B Benjamin F. Cravatt

Article Details

Volume / Issue Vol. 147, Issue 18
Published May 07, 2025
Pages 15554-15566
ISSN 0002-7863
Publisher American Chemical Society

Journal Info

Journal of the American Chemical Society

American Chemical Society

ISSN: 0002-7863 Physical Sciences

Authors (14)

H

Hayden A. Sharma

Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States

M

Michael Bielecki

Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States

M

Meredith A. Holm

Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States

T

Ty M. Thompson

Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States

Y

Yue Yin

J

Jacob B. Cravatt

Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States

T

Timothy B. Ware

Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States

A

Alex Reed

Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States

M

Molhm Nassir

T

Tamara El-Hayek Ewing

Department of Chemistry, Scripps Research, 10550 North Torrey Pines Road, La Jolla, California 92037, United States

B

Bruno Melillo

J

J. Fernando Bazan

ℏ Bioconsulting LLC

P

Phil S. Baran

B

Benjamin F. Cravatt