Potent Biological Activity by a Synthetic Cu(I) Cationophore Redistributing Intracellular Copper Pools

N Nathan Renier (Université libre de Bruxelles (ULB), Engineering of Molecular NanoSystems, Ecole Polytechnique De Bruxelles, Avenue F. Roosevelt 50, CP165/64, 1050 Brussels, Belgium) G Gianluca Weyckmans Mele (Université libre de Bruxelles (ULB), Engineering of Molecular NanoSystems, Ecole Polytechnique De Bruxelles, Avenue F. Roosevelt 50, CP165/64, 1050 Brussels, Belgium) P Pierre Lelièvre (Univ. Grenoble Alpes) M Mélanie Boeckstaens (Université libre de Bruxelles (ULB), Department of Molecular Biology, Biology of Membrane Transport Laboratory, 12 Rue des Professeurs Jeener et Brachet, 6041 Gosselies, Belgium) R Roy Lavendomme (Université libre de Bruxelles (ULB), Laboratoire de Chimie Organique, Faculty of Sciences, Avenue F. Roosevelt 50, CP160/06, 1050 Brussels, Belgium) A Akin Aydogan (Université libre de Bruxelles (ULB), Engineering of Molecular NanoSystems, Ecole Polytechnique De Bruxelles, Avenue F. Roosevelt 50, CP165/64, 1050 Brussels, Belgium) Y Yannick Dussein (Université libre de Bruxelles (ULB), Engineering of Molecular NanoSystems, Ecole Polytechnique De Bruxelles, Avenue F. Roosevelt 50, CP165/64, 1050 Brussels, Belgium) P Peggy Charbonnier (Univ. Grenoble Alpes) L Laurence Puillet Anselme (Grenoble Alpes Univ. Hospital (CHUGA)) B Benoit Chovelon (Grenoble Alpes Univ. Hospital (CHUGA)) H Hiram Castillo-Michel (European Synchrotron Radiation Facility, 71 Avenue Des Martyrs, 38000 Grenoble, France) N Nikolay Tumanov (Namur Institute of Structured Matter (NISM) and Namur Research Institute for Life Sciences (NARILIS), Department of Chemistry, University of Namur, 61 Rue de Bruxelles, 5000 Namur, Belgium) J Johan Wouters (Namur Institute of Structured Matter (NISM) and Namur Research Institute for Life Sciences (NARILIS), Department of Chemistry, University of Namur, 61 Rue de Bruxelles, 5000 Namur, Belgium) L Lucie Sancey (Univ. Grenoble Alpes (UGA)) B Benoit Busser (Univ. Grenoble Alpes (UGA)) A Anna Maria Marini (Université libre de Bruxelles (ULB), Department of Molecular Biology, Biology of Membrane Transport Laboratory, 12 Rue des Professeurs Jeener et Brachet, 6041 Gosselies, Belgium) G Giulia Veronesi (Université Grenoble Alpes, CNRS, CEA, IRIG, Laboratoire de Chimie et Biologie des Métaux, 17 rue des Martyrs, F-38000 Grenoble, France) I Ivan Jabin (Université libre de Bruxelles (ULB), Laboratoire de Chimie Organique, Faculty of Sciences, Avenue F. Roosevelt 50, CP160/06, 1050 Brussels, Belgium) A Aurélien Deniaud (Univ. Grenoble Alpes) H Hennie Valkenier (Université libre de Bruxelles (ULB), Engineering of Molecular NanoSystems, Ecole Polytechnique De Bruxelles, Avenue F. Roosevelt 50, CP165/64, 1050 Brussels, Belgium)

Article Details

Volume / Issue Vol. 148, Issue 1
Published January 14, 2026
Pages 593-604
ISSN 0002-7863
Publisher American Chemical Society

Journal Info

Journal of the American Chemical Society

American Chemical Society

ISSN: 0002-7863 Physical Sciences

Authors (20)

N

Nathan Renier

Université libre de Bruxelles (ULB), Engineering of Molecular NanoSystems, Ecole Polytechnique De Bruxelles, Avenue F. Roosevelt 50, CP165/64, 1050 Brussels, Belgium

G

Gianluca Weyckmans Mele

Université libre de Bruxelles (ULB), Engineering of Molecular NanoSystems, Ecole Polytechnique De Bruxelles, Avenue F. Roosevelt 50, CP165/64, 1050 Brussels, Belgium

P

Pierre Lelièvre

Univ. Grenoble Alpes

M

Mélanie Boeckstaens

Université libre de Bruxelles (ULB), Department of Molecular Biology, Biology of Membrane Transport Laboratory, 12 Rue des Professeurs Jeener et Brachet, 6041 Gosselies, Belgium

R

Roy Lavendomme

Université libre de Bruxelles (ULB), Laboratoire de Chimie Organique, Faculty of Sciences, Avenue F. Roosevelt 50, CP160/06, 1050 Brussels, Belgium

A

Akin Aydogan

Université libre de Bruxelles (ULB), Engineering of Molecular NanoSystems, Ecole Polytechnique De Bruxelles, Avenue F. Roosevelt 50, CP165/64, 1050 Brussels, Belgium

Y

Yannick Dussein

Université libre de Bruxelles (ULB), Engineering of Molecular NanoSystems, Ecole Polytechnique De Bruxelles, Avenue F. Roosevelt 50, CP165/64, 1050 Brussels, Belgium

P

Peggy Charbonnier

Univ. Grenoble Alpes

L

Laurence Puillet Anselme

Grenoble Alpes Univ. Hospital (CHUGA)

B

Benoit Chovelon

Grenoble Alpes Univ. Hospital (CHUGA)

H

Hiram Castillo-Michel

European Synchrotron Radiation Facility, 71 Avenue Des Martyrs, 38000 Grenoble, France

N

Nikolay Tumanov

Namur Institute of Structured Matter (NISM) and Namur Research Institute for Life Sciences (NARILIS), Department of Chemistry, University of Namur, 61 Rue de Bruxelles, 5000 Namur, Belgium

J

Johan Wouters

Namur Institute of Structured Matter (NISM) and Namur Research Institute for Life Sciences (NARILIS), Department of Chemistry, University of Namur, 61 Rue de Bruxelles, 5000 Namur, Belgium

L

Lucie Sancey

Univ. Grenoble Alpes (UGA)

B

Benoit Busser

Univ. Grenoble Alpes (UGA)

A

Anna Maria Marini

Université libre de Bruxelles (ULB), Department of Molecular Biology, Biology of Membrane Transport Laboratory, 12 Rue des Professeurs Jeener et Brachet, 6041 Gosselies, Belgium

G

Giulia Veronesi

Université Grenoble Alpes, CNRS, CEA, IRIG, Laboratoire de Chimie et Biologie des Métaux, 17 rue des Martyrs, F-38000 Grenoble, France

I

Ivan Jabin

Université libre de Bruxelles (ULB), Laboratoire de Chimie Organique, Faculty of Sciences, Avenue F. Roosevelt 50, CP160/06, 1050 Brussels, Belgium

A

Aurélien Deniaud

Univ. Grenoble Alpes

H

Hennie Valkenier

Université libre de Bruxelles (ULB), Engineering of Molecular NanoSystems, Ecole Polytechnique De Bruxelles, Avenue F. Roosevelt 50, CP165/64, 1050 Brussels, Belgium