Potent and selective SETDB1 covalent negative allosteric modulator reduces methyltransferase activity in cells
M
Mélanie Uguen
D
Devan J. Shell
M
Madhushika Silva
Y
Yu Deng
F
Fengling Li
M
Magdalena M. Szewczyk
K
Ka Yang
Y
Yani Zhao
M
Michael A. Stashko
J
Jacqueline L. Norris-Drouin
J
Jarod M. Waybright
S
Serap Beldar
J
Justin M. Rectenwald
A
Angie L. Mordant
T
Thomas S. Webb
L
Laura E. Herring
(Department of Pharmacology, University of North Carolina Metabolomics and Proteomics Core, University of North Carolina at Chapel Hill)
C
Cheryl H. Arrowsmith
S
Suzanne Ackloo
(Structural Genomics Consortium)
S
Steven P. Gygi
R
Robert K. McGinty
D
Dalia Barsyte-Lovejoy
P
Pengda Liu
L
Levon Halabelian
(Structural Genomics Consortium)
L
Lindsey I. James
K
Kenneth H. Pearce
S
Stephen V. Frye
Article Details
Journal
Nature Communications
Volume / Issue
Vol. 16, Issue 1
Published
February 24, 2025
ISSN
2041-1723
Publisher
Nature Portfolio
Authors (26)
M
Mélanie Uguen
D
Devan J. Shell
M
Madhushika Silva
Y
Yu Deng
F
Fengling Li
M
Magdalena M. Szewczyk
K
Ka Yang
Y
Yani Zhao
M
Michael A. Stashko
J
Jacqueline L. Norris-Drouin
J
Jarod M. Waybright
S
Serap Beldar
J
Justin M. Rectenwald
A
Angie L. Mordant
T
Thomas S. Webb
L
Laura E. Herring
Department of Pharmacology, University of North Carolina Metabolomics and Proteomics Core, University of North Carolina at Chapel Hill
C
Cheryl H. Arrowsmith
S
Suzanne Ackloo
Structural Genomics Consortium
S
Steven P. Gygi
R
Robert K. McGinty
D
Dalia Barsyte-Lovejoy
P
Pengda Liu
L
Levon Halabelian
Structural Genomics Consortium
L
Lindsey I. James
K
Kenneth H. Pearce
S
Stephen V. Frye
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