Overcoming Immune Checkpoint Inhibitor Resistance with Potent, Selective Dual αvβ6/8 Inhibitors Based on Engineered Lasso Peptides

A Anna Lechner (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) P Peter A. Jordan (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) G Gabriella Costa Machado da Cruz (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) J Jacob Lamson (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) J Jessica Gordon (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) B Bethany K. Okada (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) K Kelsey Anderson (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) R Rajan Chaudhari (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) C Christopher J. Rosario (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) J Jasmine Mikesell (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) S Scott A. McPhee (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States) M Mark J. Burk (Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States)

Article Details

Volume / Issue Vol. 147, Issue 36
Published September 10, 2025
Pages 32522-32536
ISSN 0002-7863
Publisher American Chemical Society

Journal Info

Journal of the American Chemical Society

American Chemical Society

ISSN: 0002-7863 Physical Sciences

Authors (12)

A

Anna Lechner

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

P

Peter A. Jordan

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

G

Gabriella Costa Machado da Cruz

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

J

Jacob Lamson

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

J

Jessica Gordon

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

B

Bethany K. Okada

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

K

Kelsey Anderson

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

R

Rajan Chaudhari

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

C

Christopher J. Rosario

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

J

Jasmine Mikesell

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

S

Scott A. McPhee

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States

M

Mark J. Burk

Lassogen, Inc., 3830 Valley Centre Drive, Suite 705-562, San Diego, California 92130, United States