On-Cell Saturation Transfer Difference NMR Spectroscopy on Ion Channels: Characterizing Negative Allosteric Modulator Binding Interactions of P2X7

S Serena Monaco (School of Chemistry, Pharmacy & Pharmacology, University of East Anglia, Norwich Research Park, Norwich NR4 7TJ, United Kingdom) J Jacob Browne (School of Chemistry, Pharmacy & Pharmacology, University of East Anglia, Norwich Research Park, Norwich NR4 7TJ, United Kingdom) M Matthew Wallace (School of Chemistry, Pharmacy & Pharmacology, University of East Anglia, Norwich Research Park, Norwich NR4 7TJ, United Kingdom) J Jesús Angulo (Instituto de Investigaciones Químicas (IIQ), CSIC − Universidad de Sevilla, Av. Américo Vespucio 49, Seville 41092, Spain) L Leanne Stokes (School of Chemistry, Pharmacy & Pharmacology, University of East Anglia, Norwich Research Park, Norwich NR4 7TJ, United Kingdom)

Article Details

Volume / Issue Vol. 147, Issue 36
Published September 10, 2025
Pages 32400-32411
ISSN 0002-7863
Publisher American Chemical Society

Journal Info

Journal of the American Chemical Society

American Chemical Society

ISSN: 0002-7863 Physical Sciences

Authors (5)

S

Serena Monaco

School of Chemistry, Pharmacy & Pharmacology, University of East Anglia, Norwich Research Park, Norwich NR4 7TJ, United Kingdom

J

Jacob Browne

School of Chemistry, Pharmacy & Pharmacology, University of East Anglia, Norwich Research Park, Norwich NR4 7TJ, United Kingdom

M

Matthew Wallace

School of Chemistry, Pharmacy & Pharmacology, University of East Anglia, Norwich Research Park, Norwich NR4 7TJ, United Kingdom

J

Jesús Angulo

Instituto de Investigaciones Químicas (IIQ), CSIC − Universidad de Sevilla, Av. Américo Vespucio 49, Seville 41092, Spain

L

Leanne Stokes

School of Chemistry, Pharmacy & Pharmacology, University of East Anglia, Norwich Research Park, Norwich NR4 7TJ, United Kingdom