Modular Synthetic Platform for the Elaboration of Fragments in Three Dimensions for Fragment-Based Drug Discovery

A Andres R. Gomez-Angel (Department of Chemistry) H Hanna F. Klein (Department of Chemistry) S Stephen Y. Yao (Department of Chemistry) J James R. Donald (Department of Chemistry) J James D. Firth (Department of Chemistry) R Rebecca Appiani (Department of Chemistry) C Cameron J. Palmer (Department of Chemistry) J Joshua Lincoln (Department of Chemistry) S Simon C. C. Lucas (Hit Discovery, Discovery Sciences, R&D, AstraZeneca, 1 Francis Crick Ave, Cambridge CB2 0AA, U.K.) L Lucia Fusani (Hit Discovery, Discovery Sciences, R&D, AstraZeneca, 1 Francis Crick Ave, Cambridge CB2 0AA, U.K.) R R. Ian Storer (Hit Discovery, Discovery Sciences, R&D, AstraZeneca, 1 Francis Crick Ave, Cambridge CB2 0AA, U.K.) P Peter O’Brien (Department of Chemistry)

Article Details

Volume / Issue Vol. 147, Issue 32
Published August 13, 2025
Pages 29292-29303
ISSN 0002-7863
Publisher American Chemical Society

Journal Info

Journal of the American Chemical Society

American Chemical Society

ISSN: 0002-7863 Physical Sciences

Authors (12)

A

Andres R. Gomez-Angel

Department of Chemistry

H

Hanna F. Klein

Department of Chemistry

S

Stephen Y. Yao

Department of Chemistry

J

James R. Donald

Department of Chemistry

J

James D. Firth

Department of Chemistry

R

Rebecca Appiani

Department of Chemistry

C

Cameron J. Palmer

Department of Chemistry

J

Joshua Lincoln

Department of Chemistry

S

Simon C. C. Lucas

Hit Discovery, Discovery Sciences, R&D, AstraZeneca, 1 Francis Crick Ave, Cambridge CB2 0AA, U.K.

L

Lucia Fusani

Hit Discovery, Discovery Sciences, R&D, AstraZeneca, 1 Francis Crick Ave, Cambridge CB2 0AA, U.K.

R

R. Ian Storer

Hit Discovery, Discovery Sciences, R&D, AstraZeneca, 1 Francis Crick Ave, Cambridge CB2 0AA, U.K.

P

Peter O’Brien

Department of Chemistry