Highly Specific Miniaturized Fluorescent Monoacylglycerol Lipase Probes Enable Translational Research

A Axel Hentsch (Leibniz Forschungsinstitut für Molekulare Pharmakologie, Campus Berlin-Buch, 13125 Berlin, Germany) M Mónica Guberman (Leibniz Forschungsinstitut für Molekulare Pharmakologie, Campus Berlin-Buch, 13125 Berlin, Germany) S Silke Radetzki (Leibniz Forschungsinstitut für Molekulare Pharmakologie, Campus Berlin-Buch, 13125 Berlin, Germany) S Sofia Kaushik (Leibniz Forschungsinstitut für Molekulare Pharmakologie, Campus Berlin-Buch, 13125 Berlin, Germany) M Mirjam Huizenga (Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research) Y Yingfang He (ETH Zürich, Institute of Pharmaceutical Sciences, Vladimir-Prelog-Weg 4, 8093 Zürich, Switzerland) J Jörg Contzen (Charité─Universitätsmedizin Berlin) B Bernd Kuhn J Jörg Benz (Roche Pharma Research & Early Development) M Maria Schippers (Roche Pharma Research & Early Development) J Jerome Paul (Leibniz Forschungsinstitut für Molekulare Pharmakologie, Campus Berlin-Buch, 13125 Berlin, Germany) L Lea Leibrock (Roche Pharma Research & Early Development) L Ludovic Collin (Roche Pharma Research & Early Development) M Matthias Wittwer (Roche Pharma Research & Early Development) A Andreas Topp (Roche Pharma Research & Early Development) F Fionn O’Hara (Roche Pharma Research & Early Development) D Dominik Heer (Roche Pharma Research & Early Development) R Remo Hochstrasser (Roche Pharma Research & Early Development) J Julie Blaising (Roche Pharma Research & Early Development) J Jens P. von Kries (Leibniz Forschungsinstitut für Molekulare Pharmakologie, Campus Berlin-Buch, 13125 Berlin, Germany) L Linjing Mu (ETH Zürich, Institute of Pharmaceutical Sciences, Vladimir-Prelog-Weg 4, 8093 Zürich, Switzerland) M Mario van der Stelt (Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research) P Philipp Mergenthaler (Charité─Universitätsmedizin Berlin) N Noa Lipstein U Uwe Grether (Roche Pharma Research & Early Development) M Marc Nazaré (Leibniz Forschungsinstitut für Molekulare Pharmakologie, Campus Berlin-Buch, 13125 Berlin, Germany)

Article Details

Volume / Issue Vol. 147, Issue 12
Published March 26, 2025
Pages 10188-10202
ISSN 0002-7863
Publisher American Chemical Society

Journal Info

Journal of the American Chemical Society

American Chemical Society

ISSN: 0002-7863 Physical Sciences

Authors (26)

A

Axel Hentsch

Leibniz Forschungsinstitut für Molekulare Pharmakologie, Campus Berlin-Buch, 13125 Berlin, Germany

M

Mónica Guberman

Leibniz Forschungsinstitut für Molekulare Pharmakologie, Campus Berlin-Buch, 13125 Berlin, Germany

S

Silke Radetzki

Leibniz Forschungsinstitut für Molekulare Pharmakologie, Campus Berlin-Buch, 13125 Berlin, Germany

S

Sofia Kaushik

Leibniz Forschungsinstitut für Molekulare Pharmakologie, Campus Berlin-Buch, 13125 Berlin, Germany

M

Mirjam Huizenga

Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research

Y

Yingfang He

ETH Zürich, Institute of Pharmaceutical Sciences, Vladimir-Prelog-Weg 4, 8093 Zürich, Switzerland

J

Jörg Contzen

Charité─Universitätsmedizin Berlin

B

Bernd Kuhn

J

Jörg Benz

Roche Pharma Research & Early Development

M

Maria Schippers

Roche Pharma Research & Early Development

J

Jerome Paul

Leibniz Forschungsinstitut für Molekulare Pharmakologie, Campus Berlin-Buch, 13125 Berlin, Germany

L

Lea Leibrock

Roche Pharma Research & Early Development

L

Ludovic Collin

Roche Pharma Research & Early Development

M

Matthias Wittwer

Roche Pharma Research & Early Development

A

Andreas Topp

Roche Pharma Research & Early Development

F

Fionn O’Hara

Roche Pharma Research & Early Development

D

Dominik Heer

Roche Pharma Research & Early Development

R

Remo Hochstrasser

Roche Pharma Research & Early Development

J

Julie Blaising

Roche Pharma Research & Early Development

J

Jens P. von Kries

Leibniz Forschungsinstitut für Molekulare Pharmakologie, Campus Berlin-Buch, 13125 Berlin, Germany

L

Linjing Mu

ETH Zürich, Institute of Pharmaceutical Sciences, Vladimir-Prelog-Weg 4, 8093 Zürich, Switzerland

M

Mario van der Stelt

Division of Drug Discovery and Safety, Leiden Academic Centre for Drug Research

P

Philipp Mergenthaler

Charité─Universitätsmedizin Berlin

N

Noa Lipstein

U

Uwe Grether

Roche Pharma Research & Early Development

M

Marc Nazaré

Leibniz Forschungsinstitut für Molekulare Pharmakologie, Campus Berlin-Buch, 13125 Berlin, Germany