GPR3 Ligands Discovered through Combined Virtual and Conformational Biosensor-Based Screening

H Hannes Schihada A Aida Shahraki (Philipps-Universität Marburg, Institute of Pharmaceutical Chemistry, Marbacher Weg 8, 35032 Marburg, Germany) A Ainoleena Turku-Metsänen (Section of Receptor Biology & Signaling, Department of Physiology and Pharmacology) M Maximilian Rath (Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, 93053 Regensburg, Germany) L Lukas Wirth (Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, 93053 Regensburg, Germany) K Katarina Nemec (Max Delbrück Center for Molecular Medicine in the Helmholtz Association) H Hrisowalantu Tselepli (Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, 93053 Regensburg, Germany) L Laura Heitzer (Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, 93053 Regensburg, Germany) B Bernadette Vallaster (Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, 93053 Regensburg, Germany) M Mariam Fadel (Philipps-Universität Marburg, Institute of Pharmaceutical Chemistry, Marbacher Weg 8, 35032 Marburg, Germany) G Gunnar Schulte D Daniel Hilger (Philipps-Universität Marburg, Institute of Pharmaceutical Chemistry, Marbacher Weg 8, 35032 Marburg, Germany) S Steffen Pockes (Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, 93053 Regensburg, Germany) M Martin J. Lohse P Peter Kolb (Philipps-Universität Marburg, Institute of Pharmaceutical Chemistry, Marbacher Weg 8, 35032 Marburg, Germany)

Article Details

Volume / Issue Vol. 148, Issue 19
Published May 20, 2026
Pages 20285-20295
ISSN 0002-7863
Publisher American Chemical Society

Journal Info

Journal of the American Chemical Society

American Chemical Society

ISSN: 0002-7863 Physical Sciences

Authors (15)

H

Hannes Schihada

A

Aida Shahraki

Philipps-Universität Marburg, Institute of Pharmaceutical Chemistry, Marbacher Weg 8, 35032 Marburg, Germany

A

Ainoleena Turku-Metsänen

Section of Receptor Biology & Signaling, Department of Physiology and Pharmacology

M

Maximilian Rath

Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, 93053 Regensburg, Germany

L

Lukas Wirth

Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, 93053 Regensburg, Germany

K

Katarina Nemec

Max Delbrück Center for Molecular Medicine in the Helmholtz Association

H

Hrisowalantu Tselepli

Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, 93053 Regensburg, Germany

L

Laura Heitzer

Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, 93053 Regensburg, Germany

B

Bernadette Vallaster

Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, 93053 Regensburg, Germany

M

Mariam Fadel

Philipps-Universität Marburg, Institute of Pharmaceutical Chemistry, Marbacher Weg 8, 35032 Marburg, Germany

G

Gunnar Schulte

D

Daniel Hilger

Philipps-Universität Marburg, Institute of Pharmaceutical Chemistry, Marbacher Weg 8, 35032 Marburg, Germany

S

Steffen Pockes

Institute of Pharmacy, University of Regensburg, Universitätsstraße 31, 93053 Regensburg, Germany

M

Martin J. Lohse

P

Peter Kolb

Philipps-Universität Marburg, Institute of Pharmaceutical Chemistry, Marbacher Weg 8, 35032 Marburg, Germany