Comprehensive Chemoproteomics Unveils Selective HMG-CoA Synthase 1 Inhibitors for Targeting Mevalonate Metabolism in Cancer

L Liang Sun S Sang Ah Yi B Brittany Q. Pham (Chemical Biology Program, Sloan Kettering Institute) A Antoine Mocellin (Cell Biology Program, Sloan Kettering Institute) S Sagnik Sen (Structural Biology Core) M M. Jason de la Cruz (Structural Biology Core) A Alban Ordureau H Heeseon An

Article Details

Volume / Issue Vol. 148, Issue 20
Published May 27, 2026
Pages 20705-20719
ISSN 0002-7863
Publisher American Chemical Society

Journal Info

Journal of the American Chemical Society

American Chemical Society

ISSN: 0002-7863 Physical Sciences

Authors (8)

L

Liang Sun

S

Sang Ah Yi

B

Brittany Q. Pham

Chemical Biology Program, Sloan Kettering Institute

A

Antoine Mocellin

Cell Biology Program, Sloan Kettering Institute

S

Sagnik Sen

Structural Biology Core

M

M. Jason de la Cruz

Structural Biology Core

A

Alban Ordureau

H

Heeseon An