Bringing Silicon to Drugs: Modular Construction of Sila-Pharmacophores for the Development of Target Protein Degraders

Z Zhigang Wu (Taizhou Research Institute) X Xujiang Zhu (Kekulé Institute of Organic Chemistry and Biochemistry, University of Bonn, Gerhard-Domagk-Straße 1, Bonn 53121, Germany) Y Yueqiu Li (Department of Chemistry) X Xia Wang M Meizhen Huang (Department of Chemistry) Z Zhenyuan Dong (Department of Chemistry) J Jiangnan Zheng (Department of Chemistry) R Ruijun Tian (Taizhou Research Institute) C Chuan He J Jie Wang (State Key Laboratory of Molecular Oncology, Beijing Key Laboratory, CAMS Key Laboratory of Translational Research on Lung Cancer, Department of Medical Oncology Cancer Hospital, Chinese Academy of Medical Sciences Beijing China)

Article Details

Volume / Issue Vol. 148, Issue 17
Published May 06, 2026
Pages 18265-18275
ISSN 0002-7863
Publisher American Chemical Society

Journal Info

Journal of the American Chemical Society

American Chemical Society

ISSN: 0002-7863 Physical Sciences

Authors (10)

Z

Zhigang Wu

Taizhou Research Institute

X

Xujiang Zhu

Kekulé Institute of Organic Chemistry and Biochemistry, University of Bonn, Gerhard-Domagk-Straße 1, Bonn 53121, Germany

Y

Yueqiu Li

Department of Chemistry

X

Xia Wang

M

Meizhen Huang

Department of Chemistry

Z

Zhenyuan Dong

Department of Chemistry

J

Jiangnan Zheng

Department of Chemistry

R

Ruijun Tian

Taizhou Research Institute

C

Chuan He

J

Jie Wang

State Key Laboratory of Molecular Oncology, Beijing Key Laboratory, CAMS Key Laboratory of Translational Research on Lung Cancer, Department of Medical Oncology Cancer Hospital, Chinese Academy of Medical Sciences Beijing China