Biosynthesis of the Red Algal Diterpene Peyssonnosol in Bacteria

Z Zhiyong Yin (Kekulé-Institute for Organic Chemistry and Biochemistry, University of Bonn, Gerhard-Domagk-Straße 1, Bonn 53121, Germany) Z Zhehui Hu (State Key Laboratory of Quantitative Engineering Biology, Shenzhen Institute of Synthetic Biology, Center of Materials Synthetic Biology) K Kexin Yang (School of Life Science and Technology, ShanghaiTech University) G Guihu Lu (State Key Laboratory of Quantitative Engineering Biology, Shenzhen Institute of Synthetic Biology, Center of Materials Synthetic Biology) G Georges B. Tabekoueng (Kekulé Institute of Organic Chemistry and Biochemistry University of Bonn Gerhard‐Domagk‐Straße 1 53121 Bonn Germany) P Pingping Wu Q Qi Luo (Guangdong Provincial Key Laboratory of Chinese Medicine Pharmaceutics, School of Traditional Chinese Medicine) J Juan Xu (Shanghai Engineering Research Center of Biotransformation of Organic Solid Waste, School of Ecological and Environmental Sciences) B Bernd Goldfuss (Institute of Organic Chemistry, Department of Chemistry, University of Cologne, Greinstraße 4, 50939 Cologne, Germany) J Jeroen S. Dickschat (Kekulé Institute for Organic Chemistry and Biochemistry, University of Bonn, Gerhard-Domagk-Straße 1, 53121 Bonn, Germany) G Guangkai Bian (State Key Laboratory of Quantitative Engineering Biology, Shenzhen Institute of Synthetic Biology, Center of Materials Synthetic Biology)

Abstract

Abstract Two diterpene synthases (DTSs) for peyssonnosol and peyssonnosol B were discovered in bacteria. Their enzyme mechanisms were investigated through isotopic labelling experiments, density functional theory (DFT) calculations and site‐directed mutagenesis, yielding biosynthetically related molecules that gave important insights into the terpene cyclisation cascade. In the present case, several mechanisms in line with the isotopic labelling experiments could be formulated. Only an extended experimental approach in combination with computational chemistry ultimately resulted in a refined mechanistic model.

Article Details

Volume / Issue Vol. 64, Issue 34
Published August 18, 2025
ISSN 1433-7851
Publisher Wiley

Journal Info

Angewandte Chemie International Edition

Wiley

ISSN: 1433-7851 Physical Sciences

Authors (11)

Z

Zhiyong Yin

Kekulé-Institute for Organic Chemistry and Biochemistry, University of Bonn, Gerhard-Domagk-Straße 1, Bonn 53121, Germany

Z

Zhehui Hu

State Key Laboratory of Quantitative Engineering Biology, Shenzhen Institute of Synthetic Biology, Center of Materials Synthetic Biology

K

Kexin Yang

School of Life Science and Technology, ShanghaiTech University

G

Guihu Lu

State Key Laboratory of Quantitative Engineering Biology, Shenzhen Institute of Synthetic Biology, Center of Materials Synthetic Biology

G

Georges B. Tabekoueng

Kekulé Institute of Organic Chemistry and Biochemistry University of Bonn Gerhard‐Domagk‐Straße 1 53121 Bonn Germany

P

Pingping Wu

Q

Qi Luo

Guangdong Provincial Key Laboratory of Chinese Medicine Pharmaceutics, School of Traditional Chinese Medicine

J

Juan Xu

Shanghai Engineering Research Center of Biotransformation of Organic Solid Waste, School of Ecological and Environmental Sciences

B

Bernd Goldfuss

Institute of Organic Chemistry, Department of Chemistry, University of Cologne, Greinstraße 4, 50939 Cologne, Germany

J

Jeroen S. Dickschat

Kekulé Institute for Organic Chemistry and Biochemistry, University of Bonn, Gerhard-Domagk-Straße 1, 53121 Bonn, Germany

G

Guangkai Bian

State Key Laboratory of Quantitative Engineering Biology, Shenzhen Institute of Synthetic Biology, Center of Materials Synthetic Biology