Abstract 5769 Selection of peptide-based and small molecule antagonists for the PAC1 receptor by combining molecular dynamics simulations and a set of biologically relevant cell-based assays
L
Lee Eiden
W
Wenqin Xu
W
Wenjuan Ye
X
Xin Hu
J
Juan Marugan
M
Mark Henderson
P
Patrick Sexton
G
Giuseppe Deganutti
Article Details
Journal
Journal of Biological Chemistry
Volume / Issue
Vol. 302, Issue 5
Published
May 01, 2026
Pages
111961
ISSN
0021-9258
Publisher
Elsevier BV
Authors (8)
L
Lee Eiden
W
Wenqin Xu
W
Wenjuan Ye
X
Xin Hu
J
Juan Marugan
M
Mark Henderson
P
Patrick Sexton
G
Giuseppe Deganutti
Related Articles from this Journal
Asialoglycoprotein receptor subunit Asgr1a loss results in attenuated cholesterol absorption in zebrafish fed a western diet
Joshua T. Derrick, Tabea O.C. Moll et al.
Aug 2026
10.1016/j.jbc.2026.113239
Nrf2-mediated epigenetic priming of osmoprotective genes enhances cellular adaptation to hyperosmotic stress
Yi Lu, Na Li et al.
Aug 2026
10.1016/j.jbc.2026.113278
Saturated cardiolipins are potent disruptors of inner mitochondrial membrane structure and function
Kailash Venkatraman, Daniel Milshteyn et al.
Aug 2026
10.1016/j.jbc.2026.113306
Epigenetic silencing of miR-141 via core promoter methylation is associated with short-term bladder cancer progression
Katerina-Marina Pilala, Artemis-Melina Papadimitriou et al.
Aug 2026
10.1016/j.jbc.2026.113302
Correction: Abstract 5588 Multifunctional carbon dots nanocarriers: Dual-drug delivery via π-π stacking interaction for stimuli-responsive chemotherapy and high oxidative stress
Girum Demissie, Jia Chang
Aug 2026
10.1016/j.jbc.2026.113253