A Tandem Bioorthogonal Retro-Cope and Cope Elimination for the Activation of Covalent Inhibitors with an Acrylamide or Vinylsulfonamide Warhead in Live Cells

Y Yan Huang M Miao Liu (Department of Genetics, Yale University School of Medicine, New Haven, CT, USA.) D Dongguang Fan F Fan Xu (CAS Key Laboratory of Colloid, Interface and Thermodynamics) F Fushuang Xiang Q Qingqiang Min X Xingyue Ji

Article Details

Volume / Issue Vol. 148, Issue 7
Published February 25, 2026
Pages 8002-8011
ISSN 0002-7863
Publisher American Chemical Society

Journal Info

Journal of the American Chemical Society

American Chemical Society

ISSN: 0002-7863 Physical Sciences

Authors (7)

Y

Yan Huang

M

Miao Liu

Department of Genetics, Yale University School of Medicine, New Haven, CT, USA.

D

Dongguang Fan

F

Fan Xu

CAS Key Laboratory of Colloid, Interface and Thermodynamics

F

Fushuang Xiang

Q

Qingqiang Min

X

Xingyue Ji