A Rare Noncoding Enhancer Variant in <i>SCN5A</i> Contributes to the High Prevalence of Brugada Syndrome in Thailand

R Roddy Walsh (Cardiovascular and Genomics Research Institute, City St. George’s, University of London, London, UK (R.W.).) J John Mauleekoonphairoj (Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.) I Isabella Mengarelli (Departments of Experimental Cardiology (R.W., I.M., F.M.B., A.O.V., M.K., L.B., C.R.B.), Amsterdam University Medical Centers, University of Amsterdam, the Netherlands.) F Fernanda M. Bosada (Departments of Experimental Cardiology (R.W., I.M., F.M.B., A.O.V., M.K., L.B., C.R.B.), Amsterdam University Medical Centers, University of Amsterdam, the Netherlands.) A Arie O. Verkerk K Karel van Duijvenboden Y Yong Poovorawan W Wanwarang Wongcharoen B Boosamas Sutjaporn (Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.) P Pharawee Wandee (Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.) N Nitinan Chimparlee (Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.) R Ronpichai Chokesuwattanaskul (Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.) K Kornkiat Vongpaisarnsin P Piyawan Dangkao (Center of Excellence in Forensic Genetics, Ratchadapiseksompotch Fund (K.V., P.D.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.) C Cheng-I Wu (Heart Rhythm Center, Division of Cardiology, Department of Medicine, Taipei Veterans General Hospital, Taiwan (C.-I.W.).) R Rafik Tadros (Research Center (S.S., P.J., S.G., I.H.-C., A.F., N.E.I., N.B., M.A., K.D., P.G.G., P.K., L.M., B.M., A.M.P., L.R., D.R., B.T., J.-C.T., J.C.-T., A.R.-P., R.T.), Montreal Heart Institute, QC, Canada.) A Ahmad S. Amin (Department of Experimental Cardiology, Amsterdam Cardiovascular Sciences, Heart Failure &amp; Arrhythmias, Amsterdam University Medical Centers, University of Amsterdam, The Netherlands (A.S.A., E.P., C.R.B.).) K Krystien V.V. Lieve (Amsterdam Cardiovascular Sciences, Heart Failure and Arrhythmias, the Netherlands (R.W., I.M., F.M.B., A.O.V., A.S.A., K.V.V.L., P.G.P., M.K., L.B., V.M.C., A.A.M.W., C.R.B.).) P Pieter G. Postema (Department of Cardiology, Amsterdam UMC, Amsterdam, The Netherlands (L.H.G.A.H., M.J.W.G., M.F.K., M.J.S., P.G.P., S.A.J.C., C.P.A., M.J.B.K.).) M Maarten Kooyman (Departments of Experimental Cardiology (R.W., I.M., F.M.B., A.O.V., M.K., L.B., C.R.B.), Amsterdam University Medical Centers, University of Amsterdam, the Netherlands.) L Leander Beekman (Departments of Experimental Cardiology (R.W., I.M., F.M.B., A.O.V., M.K., L.B., C.R.B.), Amsterdam University Medical Centers, University of Amsterdam, the Netherlands.) D Dujdao Sahasatas (Department of Medicine, Faculty of Medicine, Khon Kaen University, Thailand (D.S., P.M.).) M Montawatt Amnueypol (Departments of Medicine, Faculty of Medicine at Ramathibodi Hospital (M.A., T. Ngarmukos), Mahidol University, Bangkok, Thailand.) R Rungroj Krittayaphong S Somchai Prechawat (Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.) A Alisara Anannab (Department of Cardiovascular and Intervention, Central Chest Institute of Thailand, Nonthaburi, Thailand (A.A.).) P Pattarapong Makarawate (Department of Medicine, Faculty of Medicine, Khon Kaen University, Thailand (D.S., P.M.).) T Tachapong Ngarmukos (Departments of Medicine, Faculty of Medicine at Ramathibodi Hospital (M.A., T. Ngarmukos), Mahidol University, Bangkok, Thailand.) K Keerapa Phusanti (Department of Medicine, Maharat Nakhon Ratchasima Hospital, Nakorn Ratchasima, Thailand (K.P.).) G Gumpanart Veerakul (Bangkok Heart Hospital, Bangkok General Hospital, Thailand (G.V., A.K.).) Z Zoya Kingsbury T Taksina Newington (Illumina Cambridge Ltd, Granta Park, Great Abington, Cambridge, UK (Z.K., T. Newington, U.M., M.T.R.).) U Uma Maheswari (Illumina Cambridge Ltd, Granta Park, Great Abington, Cambridge, UK (Z.K., T. Newington, U.M., M.T.R.).) M Mark T. Ross A Andrew Grace (Department of Biochemistry, University of Cambridge, UK (A.G.).) P Pier D. Lambiase E Elijah R. Behr J Jean-Jacques Schott (Nantes Université, CHU Nantes, Centre national de la recherche scientifique, Institut national de la santé et de la recherche médicale, L’Institut du Thorax, France (A.S.B., F.L., S.L.S., F.S., C.D., T.L.T., J.-J.S.).) R Richard Redon (Nantes Université, Centre Hospitalier Universitaire (CHU) Nantes, Centre National de la Recherche Scientifique (CNRS), INSERM, l’Institut du Thorax, Nantes, France) J Julien Barc (Nantes Universite, Nantes, France) V Vincent M. Christoffels A Arthur A.M. Wilde (Heart Center, Department of Cardiology, Amsterdam Cardiovascular Sciences Heart Failure &amp; Arrhythmias, Amsterdam UMC location University of Amsterdam, Amsterdam, the Netherlands (R.E.K., L.A.D., A.-F.B.E.Q., T.F.B., A.d.W., N.R.B., W.v.d.S., J.A.d.V., K.M.K., S.P., A.A.M.W., L.R.A.O.N., L.S., L.V.A.B.).) K Koonlawee Nademanee (Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.) C Connie R. Bezzina A Apichai Khongphatthanayothin (Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.)

Abstract

BACKGROUND: Brugada syndrome (BrS) is a cardiac arrhythmia disorder that causes sudden death in young adults. Rare genetic variants in the SCN5A gene encoding the Na v 1.5 sodium channel and common noncoding variants at this locus are robustly associated with the condition. BrS is particularly prevalent in Southeast Asia but the underlying ancestry-specific factors remain largely unknown. METHODS: Genome sequencing of BrS probands and population-matched controls from Thailand was performed to identify rare noncoding variants at the SCN5A-SCN10A locus that were enriched in patients with BrS. A likely causal variant was prioritized by computational methods and introduced into human induced pluripotent stem cell (hiPSC) lines using CRISPR-Cas9. The effect of the variant on SCN5A expression and Na v 1.5 sodium channel current was then assessed in hiPSC-derived cardiomyocytes (hiPSC-CMs). RESULTS: A rare noncoding variant in an SCN5A intronic enhancer region was highly enriched in patients with BrS (detected in 3.9% of cases with a case-control odds ratio of 45.2). The variant affects a nucleotide conserved across all mammalian species and predicted to disrupt a Mef2 transcription factor binding site. Heterozygous introduction of the enhancer variant in hiPSC-CMs caused significantly reduced SCN5A expression from the variant-containing allele and a 30% reduction in Na v 1.5-mediated sodium current density compared with isogenic controls, confirming its pathogenicity. Patients with the variant had severe phenotypes, with 89% experiencing cardiac arrest. CONCLUSIONS: This is the first example of a functionally validated rare noncoding variant at the SCN5A locus and highlights how genome sequencing in understudied populations can identify novel disease mechanisms. The variant partly explains the increased prevalence of BrS in this region and enables the identification of at-risk variant carriers to reduce the burden of sudden cardiac death in Thailand.

Article Details

Journal Circulation
Volume / Issue Vol. 151, Issue 1
Published January 07, 2025
Pages 31-44
ISSN 0009-7322
Publisher Lippincott Williams & Wilkins

Journal Info

Circulation

Lippincott Williams & Wilkins

ISSN: 0009-7322 Health Sciences

Authors (45)

R

Roddy Walsh

Cardiovascular and Genomics Research Institute, City St. George’s, University of London, London, UK (R.W.).

J

John Mauleekoonphairoj

Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.

I

Isabella Mengarelli

Departments of Experimental Cardiology (R.W., I.M., F.M.B., A.O.V., M.K., L.B., C.R.B.), Amsterdam University Medical Centers, University of Amsterdam, the Netherlands.

F

Fernanda M. Bosada

Departments of Experimental Cardiology (R.W., I.M., F.M.B., A.O.V., M.K., L.B., C.R.B.), Amsterdam University Medical Centers, University of Amsterdam, the Netherlands.

A

Arie O. Verkerk

K

Karel van Duijvenboden

Y

Yong Poovorawan

W

Wanwarang Wongcharoen

B

Boosamas Sutjaporn

Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.

P

Pharawee Wandee

Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.

N

Nitinan Chimparlee

Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.

R

Ronpichai Chokesuwattanaskul

Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.

K

Kornkiat Vongpaisarnsin

P

Piyawan Dangkao

Center of Excellence in Forensic Genetics, Ratchadapiseksompotch Fund (K.V., P.D.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.

C

Cheng-I Wu

Heart Rhythm Center, Division of Cardiology, Department of Medicine, Taipei Veterans General Hospital, Taiwan (C.-I.W.).

R

Rafik Tadros

Research Center (S.S., P.J., S.G., I.H.-C., A.F., N.E.I., N.B., M.A., K.D., P.G.G., P.K., L.M., B.M., A.M.P., L.R., D.R., B.T., J.-C.T., J.C.-T., A.R.-P., R.T.), Montreal Heart Institute, QC, Canada.

A

Ahmad S. Amin

Department of Experimental Cardiology, Amsterdam Cardiovascular Sciences, Heart Failure &amp; Arrhythmias, Amsterdam University Medical Centers, University of Amsterdam, The Netherlands (A.S.A., E.P., C.R.B.).

K

Krystien V.V. Lieve

Amsterdam Cardiovascular Sciences, Heart Failure and Arrhythmias, the Netherlands (R.W., I.M., F.M.B., A.O.V., A.S.A., K.V.V.L., P.G.P., M.K., L.B., V.M.C., A.A.M.W., C.R.B.).

P

Pieter G. Postema

Department of Cardiology, Amsterdam UMC, Amsterdam, The Netherlands (L.H.G.A.H., M.J.W.G., M.F.K., M.J.S., P.G.P., S.A.J.C., C.P.A., M.J.B.K.).

M

Maarten Kooyman

Departments of Experimental Cardiology (R.W., I.M., F.M.B., A.O.V., M.K., L.B., C.R.B.), Amsterdam University Medical Centers, University of Amsterdam, the Netherlands.

L

Leander Beekman

Departments of Experimental Cardiology (R.W., I.M., F.M.B., A.O.V., M.K., L.B., C.R.B.), Amsterdam University Medical Centers, University of Amsterdam, the Netherlands.

D

Dujdao Sahasatas

Department of Medicine, Faculty of Medicine, Khon Kaen University, Thailand (D.S., P.M.).

M

Montawatt Amnueypol

Departments of Medicine, Faculty of Medicine at Ramathibodi Hospital (M.A., T. Ngarmukos), Mahidol University, Bangkok, Thailand.

R

Rungroj Krittayaphong

S

Somchai Prechawat

Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.

A

Alisara Anannab

Department of Cardiovascular and Intervention, Central Chest Institute of Thailand, Nonthaburi, Thailand (A.A.).

P

Pattarapong Makarawate

Department of Medicine, Faculty of Medicine, Khon Kaen University, Thailand (D.S., P.M.).

T

Tachapong Ngarmukos

Departments of Medicine, Faculty of Medicine at Ramathibodi Hospital (M.A., T. Ngarmukos), Mahidol University, Bangkok, Thailand.

K

Keerapa Phusanti

Department of Medicine, Maharat Nakhon Ratchasima Hospital, Nakorn Ratchasima, Thailand (K.P.).

G

Gumpanart Veerakul

Bangkok Heart Hospital, Bangkok General Hospital, Thailand (G.V., A.K.).

Z

Zoya Kingsbury

T

Taksina Newington

Illumina Cambridge Ltd, Granta Park, Great Abington, Cambridge, UK (Z.K., T. Newington, U.M., M.T.R.).

U

Uma Maheswari

Illumina Cambridge Ltd, Granta Park, Great Abington, Cambridge, UK (Z.K., T. Newington, U.M., M.T.R.).

M

Mark T. Ross

A

Andrew Grace

Department of Biochemistry, University of Cambridge, UK (A.G.).

P

Pier D. Lambiase

E

Elijah R. Behr

J

Jean-Jacques Schott

Nantes Université, CHU Nantes, Centre national de la recherche scientifique, Institut national de la santé et de la recherche médicale, L’Institut du Thorax, France (A.S.B., F.L., S.L.S., F.S., C.D., T.L.T., J.-J.S.).

R

Richard Redon

Nantes Université, Centre Hospitalier Universitaire (CHU) Nantes, Centre National de la Recherche Scientifique (CNRS), INSERM, l’Institut du Thorax, Nantes, France

J

Julien Barc

Nantes Universite, Nantes, France

V

Vincent M. Christoffels

A

Arthur A.M. Wilde

Heart Center, Department of Cardiology, Amsterdam Cardiovascular Sciences Heart Failure &amp; Arrhythmias, Amsterdam UMC location University of Amsterdam, Amsterdam, the Netherlands (R.E.K., L.A.D., A.-F.B.E.Q., T.F.B., A.d.W., N.R.B., W.v.d.S., J.A.d.V., K.M.K., S.P., A.A.M.W., L.R.A.O.N., L.S., L.V.A.B.).

K

Koonlawee Nademanee

Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.

C

Connie R. Bezzina

A

Apichai Khongphatthanayothin

Department of Medicine, Center of Excellence in Arrhythmia Research (J.M., W.W., B.S., P.W., N.C., R.C., S.P., K.N., A.K.), Faculty of Medicine, Chulalongkorn University, Bangkok, Thailand.