A monocentric analysis of ESCAT gene actionability detection in non-specific molecular profile (NSMP) endometrial cancer.

F Floriana Camarda (Fondazione Policlinico Universitario A. Gemelli, IRCCS, Division of Gynecologic Oncology, Catholic university of the Sacred Heart, Rome, Italy) L Luca Mastrantoni (Fondazione Policlinico Universitario Agostino Gemelli IRCCS, Rome, Italy) C Chiara Parrillo (Bioinformatics Research Core Facility, Gemelli Science and Technology Park (GSTeP), IRCCS Fondazione Policlinico Universitario Agostino Gemelli, Rome, Italy) T Tina Pasciuto M Marianna Manfredelli (Scientific Directorate, Fondazione Policlinico Universitario Agostino Gemelli IRCCS, Rome, Italy) R Rita Trozzi (Anna Fagotti, MD, PhD, and Rita Trozzi, MD, Fondazione Policlinico Universitario A. Gemelli-IRCCS, Rome, Italy, Università Cattolica del Sacro Cuore, Rome, Italy; Diana Giannarelli, PhD, MSc, Fondazione Policlinico Universitario A. Gemelli-IRCCS, Rome, Italy; and Giovanni Scambia, MD, Fondazione Policlinico Universitario A. Gemelli-IRCCS, Rome, Italy, Università Cattolica del Sacro Cuore, Rome, Italy) L Luciano Giaco' (Bioinformatics Research Core Facility, Gemelli Science and Technology Park (G-STeP), Fondazione Policlinico Universitario "A. Gemelli," IRCCS, Rome, Italy) F Federica Persiani (Bioinformatics Research Core Facility, Gemelli Science and Technology Park (GSTeP), IRCCS Fondazione Policlinico Universitario Agostino Gemelli, Rome, Italy) I Iolanda Mozzetta (Data Collection Research Core Facilty Gemelli Science and Technology Park (GSTeP), Fondazione Policlinico Universitario Agostino Gemelli IRCCS, Rome, Italy) A Angelo Minucci (Departmental Unit of Molecular and Genomic Diagnostics, Genomics Core Facility, Gemelli Science and Technology Park (G-STeP), Fondazione Policlinico Universitario "A. Gemelli," IRCCS, Rome, Italy) E Elisa De Paolis (Gemelli Science and Technology Park (G-STeP), Fondazione Policlinico Universitario Agostino Gemelli IRCCS, Rome, Italy) E Emanuele Perrone (Unit of Gynecologic Oncology, Department Woman and Child Health Sciences and Public Health, Fondazione Policlinico Universitario A. Gemelli Istituto di Ricovero e Cura a Carattere Scientifico) V Valentina Iacobelli (Fondazione Policlinico Universitario A. Gemelli, IRCCS, Division of Gynecologic Oncology, Catholic university of the Sacred Heart, Rome, Italy) G Gian Franco Zannoni (Gynecopathology and Breast Pathology Unit, Department of Women's, Children's and Public Health Sciences, Fondazione Policlinico Universitario A. Gemelli, IRCCS, Rome, Italy; Università Cattolica Del Sacro Cuore, Rome, Italy) F Francesco Fanfani (Unit of Gynecologic Oncology, Department Woman and Child Health Sciences and Public Health, Fondazione Policlinico Universitario A. Gemelli Istituto di Ricovero e Cura a Carattere Scientifico) G Giovanni Scambia C Camilla Nero (Gynecologic Oncology Unit, Department of Women’s and Children’s Health Sciences, Fondazione Policlinico Universitario "A. Gemelli," IRCCS, and Catholic University of the Sacred Heart, Rome, Italy)

Abstract

e17634 Background: The non-specific molecular profile (NSMP) subtype accounts for 50% of endometrial carcinoma (EC). It's a heterogeneous group of tumors, characterized by minimal cell mutations and low copy number variations, including both aggressive and clinically low-risk ECs. Methods: In January 2022 our institution launched a comprehensive cancer genome profiling (CGP) (FPG500 IRB approval 3837; NCT06020625) enrolling also EC patients. Oncogenic and likely oncogenic alterations were reported according to OncoKB and classified as Tier I-II-III according to ESCAT classification. The aim of the current analysis was to describe ESCAT gene actionability findings. Results: From January 1 st 2022 to December 31 st 2023, 253 patients with any FIGO stage, NSMP ECs were enrolled. Median age was 62 years and the most frequent histotype was endometrioid (96.9%). Estrogen receptors were positive in 94.5%. Overall, 233 patients (92%) had at least one tier III ESCAT alteration. The more frequent variants were found in PTEN (88%), PIK3CA (43%), FGFR2 (15%) and AKT1 (6%). 18% of patients had an ESR1 variant, while a KRAS G12C variant was found in 11% of patients. The majority of PTEN variants were R130X: R130G (40 pts, 17.2%), R130Q (17 pts, 7.3%) and R130* (10 pts, 4.3%). The PIK3CA's more frequently altered hotspots were H1047R (21 pts, 9.0%), E545D/K/Q/A (13 pts, 5.6%) and E542K (9 pts, 3.9%). The most frequent FGFR2 hotspot was S252W (16 pts, 6.9%). Mutually exclusive genes (p<0.05) were AKT and PTEN, PIK3CA and PIK3R1, FGFR2 with CTNNB1 and KRAS. Significant co-occurrence (p<0.05). was found between PTEN and PIK3CA and ARID1A. Considering ESCAT Tiers, the PI3K pathway was altered in 85% of patients. Conclusions: Our descriptive analysis aligns with existing literature data. Further investigation correlating survival and recurrence rates with molecular findings could unveil prognostic subgroups and potentially targetable variants.

Article Details

Volume / Issue Vol. 43, Issue 16_suppl
Published June 01, 2025
ISSN 0732-183X
Publisher Lippincott Williams & Wilkins

Journal Info

Journal of Clinical Oncology

Lippincott Williams & Wilkins

ISSN: 0732-183X Health Sciences

Authors (17)

F

Floriana Camarda

Fondazione Policlinico Universitario A. Gemelli, IRCCS, Division of Gynecologic Oncology, Catholic university of the Sacred Heart, Rome, Italy

L

Luca Mastrantoni

Fondazione Policlinico Universitario Agostino Gemelli IRCCS, Rome, Italy

C

Chiara Parrillo

Bioinformatics Research Core Facility, Gemelli Science and Technology Park (GSTeP), IRCCS Fondazione Policlinico Universitario Agostino Gemelli, Rome, Italy

T

Tina Pasciuto

M

Marianna Manfredelli

Scientific Directorate, Fondazione Policlinico Universitario Agostino Gemelli IRCCS, Rome, Italy

R

Rita Trozzi

Anna Fagotti, MD, PhD, and Rita Trozzi, MD, Fondazione Policlinico Universitario A. Gemelli-IRCCS, Rome, Italy, Università Cattolica del Sacro Cuore, Rome, Italy; Diana Giannarelli, PhD, MSc, Fondazione Policlinico Universitario A. Gemelli-IRCCS, Rome, Italy; and Giovanni Scambia, MD, Fondazione Policlinico Universitario A. Gemelli-IRCCS, Rome, Italy, Università Cattolica del Sacro Cuore, Rome, Italy

L

Luciano Giaco'

Bioinformatics Research Core Facility, Gemelli Science and Technology Park (G-STeP), Fondazione Policlinico Universitario "A. Gemelli," IRCCS, Rome, Italy

F

Federica Persiani

Bioinformatics Research Core Facility, Gemelli Science and Technology Park (GSTeP), IRCCS Fondazione Policlinico Universitario Agostino Gemelli, Rome, Italy

I

Iolanda Mozzetta

Data Collection Research Core Facilty Gemelli Science and Technology Park (GSTeP), Fondazione Policlinico Universitario Agostino Gemelli IRCCS, Rome, Italy

A

Angelo Minucci

Departmental Unit of Molecular and Genomic Diagnostics, Genomics Core Facility, Gemelli Science and Technology Park (G-STeP), Fondazione Policlinico Universitario "A. Gemelli," IRCCS, Rome, Italy

E

Elisa De Paolis

Gemelli Science and Technology Park (G-STeP), Fondazione Policlinico Universitario Agostino Gemelli IRCCS, Rome, Italy

E

Emanuele Perrone

Unit of Gynecologic Oncology, Department Woman and Child Health Sciences and Public Health, Fondazione Policlinico Universitario A. Gemelli Istituto di Ricovero e Cura a Carattere Scientifico

V

Valentina Iacobelli

Fondazione Policlinico Universitario A. Gemelli, IRCCS, Division of Gynecologic Oncology, Catholic university of the Sacred Heart, Rome, Italy

G

Gian Franco Zannoni

Gynecopathology and Breast Pathology Unit, Department of Women's, Children's and Public Health Sciences, Fondazione Policlinico Universitario A. Gemelli, IRCCS, Rome, Italy; Università Cattolica Del Sacro Cuore, Rome, Italy

F

Francesco Fanfani

Unit of Gynecologic Oncology, Department Woman and Child Health Sciences and Public Health, Fondazione Policlinico Universitario A. Gemelli Istituto di Ricovero e Cura a Carattere Scientifico

G

Giovanni Scambia

C

Camilla Nero

Gynecologic Oncology Unit, Department of Women’s and Children’s Health Sciences, Fondazione Policlinico Universitario "A. Gemelli," IRCCS, and Catholic University of the Sacred Heart, Rome, Italy