A Global Ligandability Map of Tryptoline Butynamide Stereoprobes Identifies Covalent Inhibitors of the Actin Maturation Protease
Y
Yijun Xiong
(Department of Chemistry)
C
Christopher J. Reinhardt
(Department of Chemistry)
T
Tracey Nguyen
(Vividion Therapeutics)
M
Melissa A. Hoffman
(Vividion Therapeutics)
G
Gabriel M. Simon
(Vividion Therapeutics)
B
Bruno Melillo
B
Benjamin F. Cravatt
Article Details
Volume / Issue
Vol. 148, Issue 21
Published
June 03, 2026
Pages
22077-22090
ISSN
0002-7863
Publisher
American Chemical Society
Journal Info
Journal of the American Chemical Society
American Chemical Society
ISSN: 0002-7863 Physical Sciences
Authors (7)
Y
Yijun Xiong
Department of Chemistry
C
Christopher J. Reinhardt
Department of Chemistry
T
Tracey Nguyen
Vividion Therapeutics
M
Melissa A. Hoffman
Vividion Therapeutics
G
Gabriel M. Simon
Vividion Therapeutics
B
Bruno Melillo
B
Benjamin F. Cravatt
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